How to apply anti-estrogens and prolactin inhibitors in the course of steroids?

Drugs from both groups are very useful even to the user of anabolic steroids. This refers to people who are thought to approach the construction of the healthy body of their dreams. But you need to use these helpers correctly and on time, otherwise from friends they will easily become enemies.

Very often, fans really underestimate all the pitfalls of these drugs. Meanwhile, the side effects of both the first and second, are much more dangerous and more global than the side effects of the same anabolic steroids. But completely do without them, too, will not work. So the only way out is to use them correctly.

What is aromatization?

Aromatization – the conversion of testosterone to estradiol (estrogen), or androstenedione to estrone. It occurs both naturally in the process of metabolism and when using drugs susceptible to aromatization.

Aromas are subject to:

  • Testosterone;
  • Methyltestosterone;
  • Methandrostenolone;
  • Human chorionic gonadotropin.

Boldenone also turns into estradiol, but it does not threaten side effects.

Oxymetholone exhibits estrogenic activity on its own and can easily provoke the entire set of estrogen-related troubles.

What is it fraught with? Everything is simple. Gynecomastia, excessive fluid accumulation, accelerated accumulation of fat in the most unexpected places – at the waist, hips and buttocks. Alas, a brutal man can acquire a loose ass. Well, acne.

Causes of aromatization

I will not talk about natural transformations, but let’s talk about those triggered by the use of steroids. There can be three reasons.

The first is the use of excess for a specific user dosages of aromatizing steroids. It is necessary to begin acquaintance with dangerous steroids from the minimum dosages and not to increase them until they cease to render due effect. If these steroids are taken for more than two months without a break, aromatase inhibitors become necessary.

The second reason is unhealthy liver. If you are doing everything right, and estrogenic side effects crawl all the same – go check the condition of the liver.

The third is an increased level of the enzyme aromatase in the body, or a large number of estrogen receptors in the skin, fatty layer and breasts. This is a special case, and you can get away with troubles here only in one way – to stop using aromatizing steroids once and for all.

To combat estradiol, two classes of drugs come to our aid:

  1. Aromatase inhibitors. Reduce the amount of estradiol in the body.
  2. Estrogen receptor blockers. Occupy estrogen receptors, and do not give estradiol molecules to join them and activate.
  3. Now specifically on drugs and how to use them correctly.

Aromatase Inhibitors

Mesterolone (Proviron)

Mesterolone (Proviron) is the most androgen. True, with his direct responsibilities, he does not cope very effectively. At least, it is definitely not worth using it as an anabolic or antcatabolic. But he very well inhibits (reduces) the amount of estradiol. That is, his appointment to prevent an excessive increase in the female sex hormone when using the same testosterone on the course.

Depending on the sensitivity of a particular organism and the height of steroid dosages, the working dose of Proviron is in the range of 25-50 mg per day. More than 50 mg to take does not make sense. If these doses do not work then you need to turn to more potent drugs.

There is a misconception about the complete safety of Proviron. This is not true. Being a derivative of dihydrotestosterone, it can provoke acne, hair loss on the head and their intensive growth on other parts of the body, as well as trouble with the prostate. That is why it is not necessary to be rude to dosages. Remember: Proviron is used on the course and immediately after it – in order to deal with excess estradiol.


Anastrozole is a new generation aromatase inhibitor. The best option to date. Quickly and effectively destroys extra estrogen molecules and, if you keep a proper dose, are well tolerated by the body. We use it only during the course for prophylaxis and immediately after its completion before PCT (POST-CURRENT THERAPY).

Dosage – half tablets every other day (0.5 mg). You can just keep in the nightstand on hand and when the first mucus appears, eat a pill immediately and another half a pill every other day until the unwanted symptoms disappear. After that, stop taking before the emergence of new troubles. After the course on the floor pills every other day for a period of a week to two, and only then we begin PCT.

Just remember – it is worth to overdo it with a reasonable dose – and side effects will come from the horn of plenty. This is usually depression, insomnia, lack of appetite, pain in the heart, decrease in speed and quality of thinking and memory impairment. And it is also possible problems with libido, pain in the bones and a sharp deterioration in the ratio of bad and good cholesterol. All this is due to an excessive decrease in estradiol in the body. A certain amount of the female hormone is necessary in the male body for its normal functioning. And as soon as its level falls below the permissible norm – the muscles stop growing, bone tissue is destroyed, the heart and nervous system suffers. And still the man grows dull and loses interest to the opposite sex. LetrozolLetrozol and Exemestane are the Anastrozole siblings. Aromatase inhibitors. That’s just the use of their men – amateurs is not permissible. Their action is so powerful that it cannot be controlled. By purchasing them, you risk getting everything I wrote above about the side effects of anastrozole, and in a hypertrophied form. Aminoglutethimide (Cytadren, Orimethen) . With the advent of anastrozole completely lost its relevance. Despite the powerful effect and high efficiency – has a bunch of side effects. The most dangerous is a sharp decrease in the synthesis of pregnenolone – the precursor of all steroid (cholesterol) hormones. Simply put – can cause problems with the reproductive system and the adrenal glands. Do you need it? TestolactonTestolactone is a new creation of the luminaries of pharmacology. A revolutionary tool – combining the stimulating action of gonadotropin in relation to the testicles and the powerful inhibition of aromatase. It can be used both during the course and after it before the PCT. One sad – it stands like a wing from an airplane. So for a mere mortal, this is still beyond fiction. And most importantly, remember two rules. The first is that any aromatase inhibitors are used exclusively during the steroid cycle (for the purpose of prevention) and immediately after its termination (in order to get rid of excess estradiol) before starting PCT. PCT uses ONLY estrogen receptor blockers (tamoxifen, clomiphene and thorimifen). Secondly, if the above dosages are not enough for you, then the problem is either inside of you (liver or genetic characteristics of the body), or (which happens MUCH more often) you need to reduce the dosages of flavoring steroids . And yet – if a seal has formed under one / two nipples – only tamoxifen will cope with it. Other antiestrogens may or may not help. This is already individual.

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